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Product name: Defactinib- VS 6063 | PF 04554878
Chemical name: N-methyl-4-(4-((3-(N-methylmethylsulfonamido)pyrazin-2-yl)methylamino)-5-(triflu or omethyl)pyrimidin-2-ylamino)benzamideMedchemexpress.com
MF: C20H21F3N8O3S
MW: 510.49
C AS NO: 1469988-75-7 Product: QL47
Purity: 98%
Soluble: Soluble in DMSOTAM Recep to r Inhibitor s
Description: or ally availableSecond -generation Inhibitor of focaladhesion kin ASe (FAK) and proline-richtyrosine kin ASe -2(PYK2)with anacceptablesafetypr of ileinclinicaltrials(IC50 values 0.6nMf or each kin ASe , and >100-foldgreaterselectivityf or FAK and PYK2 than f or othe r,non- target kin ASe sPubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22319597

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